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Opioids

Mitragynine solution / Kratom

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Mitragynine, an indole alkaloid, is the richest active alkaloid in the Mitragyna speciosa plant, commonly known as Kratom.

Synonyms9-methoxy CorynantheidineKratom7-Hydroxymitragynine
IUPAC3- ethyl- 1, 2, 3, 4, 6, 7, 12, 12b- octahydro- 8- methoxy- α- (methoxymethylene)- methyl ester, (αE, 2S, 3S, 12bS)- indolo[2, 3- a]quinolizine- 2- acetic acid
FormulaC23H30N2O4
Molecular weight398.495
CAS4098-40-2
Appearance no
Purity≥ 95%

Mitragynine itself acts primarily through the μ-opioid receptors, although its mitragynine-pseudoindoxyl oxidation product acts as an even more potent and selective μ-opioid agonist with less attraction to δ or κ receptors. Another alkaloid with a major contribution to the μ-opioid activity of kratom plant is the associated 7-hydroxymitragynine compound, which, while existing at the plant in much smaller quantities than mitragynine, is a much more powerful μ-opioid match participant.

Storage conditions: in a cool and dry place. Timing Mitragynine, can last up to 2 years with proper storage conditions.

Mitragynine, 100 μg/mL  $100
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Opioids

Buy O-DSMT Desmethyltramadol ( Desmetramadol ), (O-desmethyltramadol , Omnitram)

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o-dmst
Buy O-DSMT Desmethyltramadol ( Desmetramadol), (O-desmethyltramadol , Omnitram)

O-DSMT Desmetramadol Powder
Chemistry
O-Desmethyltramadol ( Desmetramadol ), or 3-(2-((dimethylamino)methyl)-1-

hydroxycyclohexyl)phenol, is an atypical synthetic opioid.

O-Desmethyltramadol bears analogies to codeine , but is not a morphine opiate opiate .

Instead, there are two rings including a cyclohexane ring which is bonded to a phenyl ring at R1.

This phenyl ring is substituted at R3 by a hydroxy (OH-) group.

This is an additional hydroxy group that is found in the same place as the cyclohexane ring.

And it is related to the phenyl ring, R1. O-DMST has a third substitution on its cyclohexane ring at R2. Here, the ring is bonded to a methyl group connected by a methylene bridge.

O-Desmethyltramadol is typical because it is found in a racemate (combination) of its stereoisomers.

Stereoisomers are two molecules that share the same chemical structure, but are three-dimensional.

chemical structure, but which are three-dimensional mirror images of each other.

Tramadol is produced as a racemate of its

two isomers because this combination is proven to be more effective.

By reversing the direction of the R2 and R1 bonds, the R and S enantiomers of O-Desmethyltramadol are obtained.

O-DMST is nearly identical to tramadol and is so named due to the absence of the methoxy R3 substitute for tramadol.

Price:
O-DSMT (O-desmethyltramadol , Omnitram) 10g $250
O-DSMT (O-desmethyltramadol , Omnitram) 50g $850
O-DSMT (O-desmethyltramadol , Omnitram) 100g $1050
O-DSMT (O-desmethyltramadol , Omnitram) 500g $3700
O-DSMT (O-desmethyltramadol , Omnitram) 1kg $5500

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Opioids

Buy Fentanyl Hcl

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Buy Fentanyl Hcl Powder & Crystals Online | Fentanyl Hcl Crystals & Powder For Sale

Fentanyl HCL(Intravenous) is often used for anesthesia and to treat pain. To induce anesthesia, it is given with a sedative-hypnotic, like propofol or thiopental, and a muscle relaxant. To maintain anesthesia, inhaled anesthetics and additional fentanyl may be used. These are often given in 15–30-minute intervals throughout procedures such as endoscopy, surgeries, and emergency rooms.

For pain relief after surgery, use can decrease the amount of inhalational anesthetic needed for emergence from anesthesia. Balancing this medication and titrating the drug based on expected stimuli and the person’s responses can result in stable blood pressure and heart rate throughout a procedure and a faster emergence from anesthesia with minimal pain.

2). Obstetrics
Fentanyl HCL is sometimes given intrathecally as part of spinal anesthesia or epidurally for epidural anesthesia and analgesia. Because of fentanyl’s high lipid solubility, its effects are more localized than morphine, and some clinicians prefer to use morphine to get a wider spread of analgesia. However, it is widely used in obstetrical anesthesia because of its short time to action peak (about 5 min), the rapid termination of its effect after a single dose, and the occurrence of relative cardiovascular stability.

In obstetrics, the dose must be closely regulated in order to prevent large amounts of transfer from mother to fetus. At high doses, the drug may act on the fetus to cause postnatal respiratory distress. For this reason, shorter-acting agents such as alfentanyl or remifentanil may be more suitable in the context of inducing general anesthesia.

3). Pain management
The bioavailability of intranasal fentanyl is about 70–90%, but with some imprecision due to clotted nostrils, pharyngeal swallow, and incorrect administration. For both emergency and palliative use, intranasal fentanyl is available in doses of 50, 100, and 200 µg. In emergency medicine, safe administration of intranasal fentanyl with a low rate of side effects and a promising pain-reducing effect was demonstrated in a prospective observational study in about 900 out-of-hospital patients.

In children, intranasal fentanyl is useful for the treatment of moderate and severe pain and is well tolerated.

Adverse effects
Fentanyl HCL’s most common side effects, which affect more than 10% of people, include diarrhea, nausea, constipation, dry mouth, somnolence, confusion, asthenia (weakness), sweating. Less frequently, in 3-10% of people, fentanyl can cause abdominal pain, headache, fatigue, anorexia and weight loss, dizziness, nervousness, hallucinations, anxiety, depression, flu-like symptoms, dyspepsia (indigestion), shortness of breath, hypoventilation, apnoea, and urinary retention.

Fentanyl HCL use has also been associated with aphasia. Despite being a more potent analgesic, fentanyl tends to induce less nausea, as well as less histamine-mediated itching, than morphine.

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Fentanyl Hcl 10g $350
Fentanyl Hcl 50g $1200
Fentanyl Hcl 100g $1900
Fentanyl Hcl 500g $6000
Fentanyl Hcl 1kg $9999

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Opioids

Buy Piperidinohton ( Piperidylthiambutene ) Powder

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Buy Piperidylthiambutene Powder & Crystals | Piperidinohton Crystals & Powder For Sale

Piperidinohton (Piperidylthiambutene)

Piperidinohton, also called Piperidylthiambutene, is a new opioid that has excellent analgesic properties. Piperidinohton has an efficacy equal to morphine and can show a high affinity for the μ-opioid receptor. Attention! Piperidinohton (Piperidylthiambutene) is a controlled substance in a number of countries such as the USA, Australia, New Zealand.Piperidinohton (Piperidylthiambutene)

Synonyms  Piperidinohton  Piperidylthiambutene
IUPAC 1-[4,4-Di(2-thienyl)-3-buten-2-yl]piperidin
Formula C17H21NS2
Molecular weight 303.485 g/mol
CAS 54160-31-5
Appearance Powder
Purity≥ 98%

Piperidinohton and all other synthetic opioids sold on this website are for research and legal applications. Piperidinohton is a designer drug with obvious physiological and psychoactive effects.

Side effects from Piperidinohton are not known.

Storage conditions: in a cool and dry place. Terms Piperidinohton , can last up to 2 years with proper storage conditions.  

Price :

Piperidinohton 10g $275
Piperidinohton 50g $690
Piperidinohton 100g $800
Piperidinohton 500g $2500
Piperidinohton 1kg $3900

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